1.Jingjing Peng, Chunpu Li, Mirzadavlat Khamrakulov, Jiang Wang,* and Hong Liu.* Rhodium(III)-Catalyzed C-H Alkenylation: Access to Maleimide-Decorated Tryptophan and Tryptophan-Containing Peptides. Org. Lett. 2020, 22, 1535-1541.
2.Xingjun Li, # Jiang Wang, # Xiong Xie, Wenhao Dai, Xu Han, Kaixian Chen,* Hong Liu.* Ir(III)-Catalyzed direct C-H functionalization of N-phenylacetamide with α-diazo quinones: a novel strategy for producing 2-hydroxy-2’-amino-1,2’-biaryl scaffolds. Chem. Commun. 2020, 56, 3441-3444.
3.Zunyun Fu, Xutong Li, Zhaohui Wang, Zhaojun Li, Xiaohong Liu, Xiaolong Wu, Jihui Zhao, Xiaoyu Ding, Xiaozhe Wan, Feisheng Zhong, Dingyan Wang, Xiaomin Luo, Kaixian Chen, Hong Liu, Jiang Wang,* Hualiang Jiang, Mingyue Zheng.* Optimizing Chemical Reaction Conditions Using Deep Learning: a Case Study for Suzuki-Miyaura Cross-Coupling Reactio. Org. Chem. Front., 2020, accepted.
4.Zhaohui Wang, Yangjie Fu, Qiyu Zhang, Hong Liu,* and Jiang Wang.* Pd(II)-Catalyzed Direct γ?C(sp3)?H Arylation between Free β2?Amino Esters and β3?Amino Esters and Aryl Iodides Using a Catalytic Transient Directing Group. J. Org. Chem., 2020, 85, 7683-7693.
5.Chenglin Wu,# Cong Xi,# Junhua Tong, Jing Zhao, Hualiang Jiang, Jiang Wang,* Yiping Wang,* and Hong Liu.* Design, synthesis, and biological evaluation of novel tetrahydroprotoberberine derivatives (THPBs) as proprotein convertase subtilisin/kexin type 9 (PCSK9) modulators for the treatment of hyperlipidemia. Acta Pharmaceutica Sinica B, 2019, 9, 1216-1230. (Cover)
6.Huihui Li, Chenglin Wu, Hong Liu,* and Jiang Wang.* Ruthenium(II)-Catalyzed C–H Acylmethylation between (Hetero)arenes and α-Cl Ketones/Sulfoxonium Ylides. J. Org. Chem. 2019, 84, 13262-13275.
7.Jiang Wang, # Mingbo Su, # Tingting Li, # Anhui Gao, Wei Yang, Li Sheng, Yi Zang, Jia Li,* Hong Liu.* Design, Synthesis and Biological Evaluation of Thienopyrimidine Hydroxamic Acid Based Derivatives as Structurally Novel Histone Deacetylase (HDAC) Inhibitors. Eur. J. Med. Chem. 2017, 128, 293-299.
8.Jiang Wang, Maria Sanchez-Rosello, Jose Luis Acena, Carlos del Pozo, Alexander E. Sorochinsky, Santos Fustero,* Vadim A. Soloshonok,* Hong Liu.* Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001-2011). Chem. Rev. 2014, 114, 2432-2506.
9.Xun Ji#, Mingbo Su#, Jiang Wang#, Guanghui Deng, Sisi Deng, Zeng Li, Chunlan Tang, Jingya Li, Jia Li,* Linxiang Zhao, Hualiang Jiang, Hong Liu.* Design, synthesis and biological evaluation of hetero-aromatic moieties substituted pyrrole-2-carbonitrile derivatives as dipeptidyl peptidase IV inhibitors. Eur. J. Med. Chem. 2014, 75, 111-122.
10.Jiang Wang, Shengbin Zhou, Daizong Lin, Xiao Ding, Hualiang Jiang, Hong Liu.* Highly Diastereo- and Enantioselective Synthesis of syn-β-Substituted Tryptophans via Asymmetric Michael Addition of a Chiral Equivalent of Nucleophilic Glycine and Sulfonylindoles. Chem. Commun. 2011, 47, 8355-8357. |